Drug Metabolism and Pharmacokinetics Quick Guide covers a number of aspects of drug assessment at drug discovery and development stages, topics such as pharmacokinetics, absorption, metabolism, enzyme kinetics, drug transporters, drug interactions, drug-like properties, assays and in silico calculations. It covers key concepts, with useful tables on physiological parameters (eg. blood flow to organs in x-species, expression and localization of enzymes and transporters), chemical structure, nomenclature, and moieties leading to bioactivation (with examples). Overall it includes a number of key topics useful at the drug discovery stage, which would serve as a quick reference with several examples from the literature to illustrate the concept.
| Author: Siamak Cyrus Khojasteh |
| Publisher: Springer |
| Publication Date: Apr 19, 2011 |
| Number of Pages: 214 pages |
| Binding: Paperback or Softback |
| ISBN-10: 144195628X |
| ISBN-13: 9781441956286 |